Purinergic P2X3 heteroreceptors enhance parasympathetic motor drive in isolated porcine detrusor, a reliable model for development of P2X selective blockers for detrusor hyperactivity.
D'Agostino, Gianluigi
Purinergic P2X3 heteroreceptors enhance parasympathetic motor drive in isolated porcine detrusor, a reliable model for development of P2X selective blockers for detrusor hyperactivity. [electronic resource] - Pharmacological research Jan 2012 - 129-36 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1096-1186
10.1016/j.phrs.2011.10.002 doi
Acetylcholine--metabolism
Adenosine Triphosphate--metabolism
Animals
Dose-Response Relationship, Drug
Electric Stimulation
Hydrolysis
In Vitro Techniques
Motor Neurons--drug effects
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Parasympathetic Nervous System--drug effects
Purinergic P2X Receptor Antagonists--pharmacology
Receptors, Purinergic P2X3--drug effects
Swine
Synaptic Transmission--drug effects
Time Factors
Urinary Bladder--drug effects
Urinary Bladder, Overactive--drug therapy
Purinergic P2X3 heteroreceptors enhance parasympathetic motor drive in isolated porcine detrusor, a reliable model for development of P2X selective blockers for detrusor hyperactivity. [electronic resource] - Pharmacological research Jan 2012 - 129-36 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1096-1186
10.1016/j.phrs.2011.10.002 doi
Acetylcholine--metabolism
Adenosine Triphosphate--metabolism
Animals
Dose-Response Relationship, Drug
Electric Stimulation
Hydrolysis
In Vitro Techniques
Motor Neurons--drug effects
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Parasympathetic Nervous System--drug effects
Purinergic P2X Receptor Antagonists--pharmacology
Receptors, Purinergic P2X3--drug effects
Swine
Synaptic Transmission--drug effects
Time Factors
Urinary Bladder--drug effects
Urinary Bladder, Overactive--drug therapy