Synthesis and preliminary evaluation of amiloride analogs as inhibitors of the urokinase-type plasminogen activator (uPA).

Matthews, Hayden

Synthesis and preliminary evaluation of amiloride analogs as inhibitors of the urokinase-type plasminogen activator (uPA). [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2011 - 6760-6 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2011.09.044 doi


Amiloride--analogs & derivatives
Antineoplastic Agents--chemical synthesis
Diuretics--chemical synthesis
Humans
Models, Molecular
Neoplasms--drug therapy
Structure-Activity Relationship
Urokinase-Type Plasminogen Activator--antagonists & inhibitors