Metabolism and pharmacokinetic studies of JPH203, an L-amino acid transporter 1 (LAT1) selective compound.

Wempe, Michael F

Metabolism and pharmacokinetic studies of JPH203, an L-amino acid transporter 1 (LAT1) selective compound. [electronic resource] - Drug metabolism and pharmacokinetics 2012 - 155-61 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1880-0920

10.2133/dmpk.dmpk-11-rg-091 doi


Acetylation
Animals
Antineoplastic Agents--analysis
Benzoxazoles--analysis
Biotransformation
Dogs
Humans
Intestine, Small--metabolism
Kidney--chemistry
Large Neutral Amino Acid-Transporter 1--chemistry
Liver--chemistry
Macaca fascicularis
Male
Membrane Transport Modulators--analysis
Mice
Microsomes--metabolism
Microsomes, Liver--metabolism
Rats
Rats, Sprague-Dawley
Tissue Distribution
Tyrosine--analogs & derivatives