Biochemistry and biology of 2'-Fluoro-2'-deoxythymidine (FT), a putative highly selective substrate for thymidine kinase type 2 (TK2).
Wiebe, Leonard I
Biochemistry and biology of 2'-Fluoro-2'-deoxythymidine (FT), a putative highly selective substrate for thymidine kinase type 2 (TK2). [electronic resource] - Current radiopharmaceuticals Jan 2012 - 38-46 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1874-4729
10.2174/1874471011205010038 doi
Animals
Antineoplastic Agents--pharmacology
Autoradiography
Bone Neoplasms--drug therapy
Cell Line, Tumor
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Humans
Inhibitory Concentration 50
Membrane Transport Proteins--metabolism
Mice
Mice, Inbred BALB C
Neoplasm Transplantation
Osteosarcoma--drug therapy
Phosphorylation
Positron-Emission Tomography
Radiopharmaceuticals
Thymidine--analogs & derivatives
Thymidine Kinase
Transgenes
Biochemistry and biology of 2'-Fluoro-2'-deoxythymidine (FT), a putative highly selective substrate for thymidine kinase type 2 (TK2). [electronic resource] - Current radiopharmaceuticals Jan 2012 - 38-46 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1874-4729
10.2174/1874471011205010038 doi
Animals
Antineoplastic Agents--pharmacology
Autoradiography
Bone Neoplasms--drug therapy
Cell Line, Tumor
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Humans
Inhibitory Concentration 50
Membrane Transport Proteins--metabolism
Mice
Mice, Inbred BALB C
Neoplasm Transplantation
Osteosarcoma--drug therapy
Phosphorylation
Positron-Emission Tomography
Radiopharmaceuticals
Thymidine--analogs & derivatives
Thymidine Kinase
Transgenes