Modulation of CCAAT/enhancer binding protein homologous protein (CHOP)-dependent DR5 expression by nelfinavir sensitizes glioblastoma multiforme cells to tumor necrosis factor-related apoptosis-inducing ligand (TRAIL).

Tian, Xiaobing

Modulation of CCAAT/enhancer binding protein homologous protein (CHOP)-dependent DR5 expression by nelfinavir sensitizes glioblastoma multiforme cells to tumor necrosis factor-related apoptosis-inducing ligand (TRAIL). [electronic resource] - The Journal of biological chemistry Aug 2011 - 29408-29416 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1083-351X

10.1074/jbc.M110.197665 doi


Activating Transcription Factor 4--genetics
Apoptosis--drug effects
Cell Line, Tumor
Gene Expression Regulation, Neoplastic--drug effects
Glioblastoma--drug therapy
HIV Protease Inhibitors--pharmacology
Humans
Nelfinavir--pharmacology
Neoplasm Proteins--genetics
Receptors, TNF-Related Apoptosis-Inducing Ligand--biosynthesis
TNF-Related Apoptosis-Inducing Ligand--pharmacology
Transcription Factor CHOP--genetics
Unfolded Protein Response--drug effects