Synthesis and structure-activity relationship of new 1,5-dialkyl-1,5-benzodiazepines as cholecystokinin-2 receptor antagonists.

Roberts, Karen

Synthesis and structure-activity relationship of new 1,5-dialkyl-1,5-benzodiazepines as cholecystokinin-2 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry Jul 2011 - 4257-73 p. digital

Publication Type: Journal Article

1464-3391

10.1016/j.bmc.2011.05.057 doi


Animals
Benzodiazepinones--chemical synthesis
Dogs
Guinea Pigs
Mice
Molecular Structure
Rats
Receptor, Cholecystokinin B--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship
Tissue Distribution