Effects of oral curcumin on the pharmacokinetics of intravenous and oral etoposide in rats: possible role of intestinal CYP3A and P-gp inhibition by curcumin.

Lee, Chong-Ki

Effects of oral curcumin on the pharmacokinetics of intravenous and oral etoposide in rats: possible role of intestinal CYP3A and P-gp inhibition by curcumin. [electronic resource] - Biopharmaceutics & drug disposition May 2011 - 245-51 p. digital

Publication Type: Journal Article

1099-081X

10.1002/bdd.754 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Administration, Oral
Animals
Antineoplastic Agents--administration & dosage
Antineoplastic Agents, Phytogenic--administration & dosage
Curcumin--administration & dosage
Cytochrome P-450 CYP3A--physiology
Cytochrome P-450 CYP3A Inhibitors
Drug Interactions
Etoposide--administration & dosage
Fluorescent Dyes--pharmacokinetics
Injections, Intravenous
Intestinal Mucosa--metabolism
Intestines--drug effects
Male
Rats
Rats, Sprague-Dawley
Rhodamine 123--pharmacokinetics