The discovery of potent and long-acting oral factor Xa inhibitors with tetrahydroisoquinoline and benzazepine P4 motifs.

Watson, Nigel S

The discovery of potent and long-acting oral factor Xa inhibitors with tetrahydroisoquinoline and benzazepine P4 motifs. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2011 - 1588-92 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2011.01.129 doi


Administration, Oral
Animals
Benzazepines--administration & dosage
Crystallography, X-Ray
Drug Evaluation, Preclinical
Factor Xa Inhibitors
Molecular Structure
Rats
Serine Proteinase Inhibitors--administration & dosage
Tetrahydroisoquinolines--administration & dosage