Linkage with cathepsin B-sensitive dipeptide promotes the in vitro and in vivo anticancer activity of PEGylated tumor necrosis factor-alpha (TNF-α) against murine fibrosarcoma.
Dai, ChuanYun
Linkage with cathepsin B-sensitive dipeptide promotes the in vitro and in vivo anticancer activity of PEGylated tumor necrosis factor-alpha (TNF-α) against murine fibrosarcoma. [electronic resource] - Science China. Life sciences Feb 2011 - 128-38 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1869-1889
10.1007/s11427-010-4124-z doi
Animals
Antineoplastic Agents--metabolism
Cathepsin B--antagonists & inhibitors
Cell Line, Tumor
Dipeptides--metabolism
Drug Carriers--metabolism
Female
Fibrosarcoma--drug therapy
Humans
Mice
Mice, Inbred BALB C
Microsomes, Liver--metabolism
Polyethylene Glycols--metabolism
Prodrugs--metabolism
Rats
Rats, Sprague-Dawley
Tumor Necrosis Factor-alpha--metabolism
Linkage with cathepsin B-sensitive dipeptide promotes the in vitro and in vivo anticancer activity of PEGylated tumor necrosis factor-alpha (TNF-α) against murine fibrosarcoma. [electronic resource] - Science China. Life sciences Feb 2011 - 128-38 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1869-1889
10.1007/s11427-010-4124-z doi
Animals
Antineoplastic Agents--metabolism
Cathepsin B--antagonists & inhibitors
Cell Line, Tumor
Dipeptides--metabolism
Drug Carriers--metabolism
Female
Fibrosarcoma--drug therapy
Humans
Mice
Mice, Inbred BALB C
Microsomes, Liver--metabolism
Polyethylene Glycols--metabolism
Prodrugs--metabolism
Rats
Rats, Sprague-Dawley
Tumor Necrosis Factor-alpha--metabolism