Discovery of orally available tetrahydroquinoline-based glucocorticoid receptor agonists.

Hudson, Andrew R

Discovery of orally available tetrahydroquinoline-based glucocorticoid receptor agonists. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2011 - 1697-700 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2011.01.093 doi


Administration, Oral
Animals
Drug Discovery
Enzyme-Linked Immunosorbent Assay
Humans
Quinolines--administration & dosage
Rats
Rats, Sprague-Dawley
Receptors, Glucocorticoid--agonists
Structure-Activity Relationship