3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: hit to lead studies.

Gilbert, Adam M

3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: hit to lead studies. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2011 - 195-9 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2010.11.038 doi


Allosteric Regulation
Animals
Anxiety Disorders--drug therapy
Benzamides--chemistry
Disease Models, Animal
High-Throughput Screening Assays
Mice
Pyridines--chemistry
Rats
Receptor, Metabotropic Glutamate 5
Receptors, Metabotropic Glutamate--chemistry