3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: hit to lead studies.
Gilbert, Adam M
3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: hit to lead studies. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2011 - 195-9 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2010.11.038 doi
Allosteric Regulation
Animals
Anxiety Disorders--drug therapy
Benzamides--chemistry
Disease Models, Animal
High-Throughput Screening Assays
Mice
Pyridines--chemistry
Rats
Receptor, Metabotropic Glutamate 5
Receptors, Metabotropic Glutamate--chemistry
3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: hit to lead studies. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2011 - 195-9 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2010.11.038 doi
Allosteric Regulation
Animals
Anxiety Disorders--drug therapy
Benzamides--chemistry
Disease Models, Animal
High-Throughput Screening Assays
Mice
Pyridines--chemistry
Rats
Receptor, Metabotropic Glutamate 5
Receptors, Metabotropic Glutamate--chemistry