Pharmacokinetics and pharmacodynamics of single rising intravenous doses (0.5 mg-10 mg) and determination of absolute bioavailability of the dipeptidyl peptidase-4 inhibitor linagliptin (BI 1356) in healthy male subjects.
Retlich, Silke
Pharmacokinetics and pharmacodynamics of single rising intravenous doses (0.5 mg-10 mg) and determination of absolute bioavailability of the dipeptidyl peptidase-4 inhibitor linagliptin (BI 1356) in healthy male subjects. [electronic resource] - Clinical pharmacokinetics Dec 2010 - 829-40 p. digital
Publication Type: Comparative Study; Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
1179-1926
10.2165/11536620-000000000-00000 doi
Adolescent
Adult
Area Under Curve
Biological Availability
Cross-Over Studies
Dipeptidyl Peptidase 4--metabolism
Dipeptidyl-Peptidase IV Inhibitors--administration & dosage
Dose-Response Relationship, Drug
Half-Life
Humans
Infusions, Intravenous
Linagliptin
Male
Middle Aged
Models, Biological
Protein Binding
Purines--administration & dosage
Quinazolines--administration & dosage
Single-Blind Method
Tablets
Tissue Distribution
Young Adult
Pharmacokinetics and pharmacodynamics of single rising intravenous doses (0.5 mg-10 mg) and determination of absolute bioavailability of the dipeptidyl peptidase-4 inhibitor linagliptin (BI 1356) in healthy male subjects. [electronic resource] - Clinical pharmacokinetics Dec 2010 - 829-40 p. digital
Publication Type: Comparative Study; Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
1179-1926
10.2165/11536620-000000000-00000 doi
Adolescent
Adult
Area Under Curve
Biological Availability
Cross-Over Studies
Dipeptidyl Peptidase 4--metabolism
Dipeptidyl-Peptidase IV Inhibitors--administration & dosage
Dose-Response Relationship, Drug
Half-Life
Humans
Infusions, Intravenous
Linagliptin
Male
Middle Aged
Models, Biological
Protein Binding
Purines--administration & dosage
Quinazolines--administration & dosage
Single-Blind Method
Tablets
Tissue Distribution
Young Adult