CYP4F enzymes are responsible for the elimination of fingolimod (FTY720), a novel treatment of relapsing multiple sclerosis.
Jin, Yi
CYP4F enzymes are responsible for the elimination of fingolimod (FTY720), a novel treatment of relapsing multiple sclerosis. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Feb 2011 - 191-8 p. digital
Publication Type: Journal Article
1521-009X
10.1124/dmd.110.035378 doi
Aryl Hydrocarbon Hydroxylases--genetics
Biotransformation
Chromatography, High Pressure Liquid
Cytochrome P-450 Enzyme System--genetics
Cytochrome P450 Family 4
Fingolimod Hydrochloride
Humans
In Vitro Techniques
Mass Spectrometry
Microsomes, Liver--metabolism
Molecular Structure
Multiple Sclerosis, Relapsing-Remitting--drug therapy
Oxidation-Reduction
Propylene Glycols--chemistry
Sphingosine--analogs & derivatives
Transfection
CYP4F enzymes are responsible for the elimination of fingolimod (FTY720), a novel treatment of relapsing multiple sclerosis. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Feb 2011 - 191-8 p. digital
Publication Type: Journal Article
1521-009X
10.1124/dmd.110.035378 doi
Aryl Hydrocarbon Hydroxylases--genetics
Biotransformation
Chromatography, High Pressure Liquid
Cytochrome P-450 Enzyme System--genetics
Cytochrome P450 Family 4
Fingolimod Hydrochloride
Humans
In Vitro Techniques
Mass Spectrometry
Microsomes, Liver--metabolism
Molecular Structure
Multiple Sclerosis, Relapsing-Remitting--drug therapy
Oxidation-Reduction
Propylene Glycols--chemistry
Sphingosine--analogs & derivatives
Transfection