Design and synthesis of a new class of malonyl-CoA decarboxylase inhibitors with anti-obesity and anti-diabetic activities.

Tang, Haifeng

Design and synthesis of a new class of malonyl-CoA decarboxylase inhibitors with anti-obesity and anti-diabetic activities. [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2010 - 6088-92 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2010.08.047 doi


Animals
Anti-Obesity Agents--chemical synthesis
Blood Glucose--drug effects
Body Weight--drug effects
Carboxy-Lyases--antagonists & inhibitors
Diabetes Mellitus, Type 2--drug therapy
Drug Design
Eating--drug effects
Humans
Hypoglycemic Agents--chemical synthesis
Mice
Mice, Inbred C57BL
Obesity--drug therapy
Propanols--chemical synthesis
Thiazoles--chemical synthesis