Spiroindolones, a potent compound class for the treatment of malaria.

Rottmann, Matthias

Spiroindolones, a potent compound class for the treatment of malaria. [electronic resource] - Science (New York, N.Y.) Sep 2010 - 1175-80 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1095-9203

10.1126/science.1193225 doi


Adenosine Triphosphatases--antagonists & inhibitors
Animals
Antimalarials--administration & dosage
Cell Line
Drug Discovery
Drug Resistance
Erythrocytes--parasitology
Female
Genes, Protozoan
Humans
Indoles--administration & dosage
Malaria--drug therapy
Male
Mice
Models, Molecular
Mutant Proteins--antagonists & inhibitors
Mutation
Parasitic Sensitivity Tests
Plasmodium berghei--drug effects
Plasmodium falciparum--drug effects
Plasmodium vivax--drug effects
Protein Synthesis Inhibitors--administration & dosage
Protozoan Proteins--biosynthesis
Rats
Rats, Wistar
Spiro Compounds--administration & dosage