N-tetrahydrothiochromenoisoxazole-1-carboxamides as selective antagonists of cloned human 5-HT2B.

Kwon, Yoon Jin

N-tetrahydrothiochromenoisoxazole-1-carboxamides as selective antagonists of cloned human 5-HT2B. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2010 - 5488-90 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1464-3405

10.1016/j.bmcl.2010.07.074 doi


Heterocyclic Compounds, 3-Ring--chemistry
Humans
Receptor, Serotonin, 5-HT2B--metabolism
Serotonin 5-HT2 Receptor Antagonists--chemistry
Structure-Activity Relationship