Calcimimetic R-568 effects on activity of R990G polymorphism of calcium-sensing receptor.

Terranegra, Annalisa

Calcimimetic R-568 effects on activity of R990G polymorphism of calcium-sensing receptor. [electronic resource] - Journal of molecular endocrinology Oct 2010 - 245-56 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1479-6813

10.1677/JME-10-0034 doi


Amino Acid Substitution--genetics
Aniline Compounds--pharmacology
Calcium--metabolism
Calcium Signaling--drug effects
Enzyme Activators--pharmacology
Extracellular Signal-Regulated MAP Kinases--metabolism
HEK293 Cells
Humans
Phenethylamines
Phosphorylation--drug effects
Polymorphism, Single Nucleotide--genetics
Propylamines
Protein Kinase C--antagonists & inhibitors
Protein Kinase Inhibitors--pharmacology
Receptors, Calcium-Sensing--genetics
Sarcoplasmic Reticulum Calcium-Transporting ATPases--antagonists & inhibitors
Signal Transduction--drug effects
Type C Phospholipases--antagonists & inhibitors