Pyrrolo[1,2-a]pyrazine and pyrazolo[1,5-a]pyrazine: novel, potent, and selective series of Vasopressin 1b receptor antagonists.

Arban, Roberto

Pyrrolo[1,2-a]pyrazine and pyrazolo[1,5-a]pyrazine: novel, potent, and selective series of Vasopressin 1b receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2010 - 5044-9 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2010.07.037 doi


Antidiuretic Hormone Receptor Antagonists
Pyrazines--chemistry
Pyrroles--chemistry
Structure-Activity Relationship