Non-stereo-selective cytosolic human brain tissue 3-ketosteroid reductase is refractory to inhibition by AKR1C inhibitors.

Steckelbroeck, Stephan

Non-stereo-selective cytosolic human brain tissue 3-ketosteroid reductase is refractory to inhibition by AKR1C inhibitors. [electronic resource] - Biochimica et biophysica acta Nov 2010 - 1221-31 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

0006-3002

10.1016/j.bbalip.2010.07.005 doi


20-Hydroxysteroid Dehydrogenases--antagonists & inhibitors
3-Hydroxysteroid Dehydrogenases--metabolism
Adult
Aged
Brain--metabolism
Cell Line, Tumor
Chromatography, Thin Layer--methods
Female
Gas Chromatography-Mass Spectrometry--methods
Gene Expression Regulation, Enzymologic
Humans
Infant
Middle Aged
Steroid 17-alpha-Hydroxylase--genetics
Steroids--chemistry
Temporal Lobe--pathology