Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805.
Baffert, Fabienne
Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805. [electronic resource] - Molecular cancer therapeutics Jul 2010 - 1945-55 p. digital
Publication Type: Journal Article
1538-8514
10.1158/1535-7163.MCT-10-0053 doi
Adenosine Triphosphate--pharmacology
Animals
Apoptosis--drug effects
Cell Line
Cell Line, Tumor
Cell Proliferation--drug effects
Erythropoiesis--drug effects
Humans
Janus Kinase 2--antagonists & inhibitors
K562 Cells
Mice
Mice, Inbred BALB C
Mice, SCID
Models, Molecular
Molecular Structure
Mutation
Phosphorylation--drug effects
Polycythemia--metabolism
Protein Structure, Tertiary
Quinoxalines--chemistry
Rats
STAT5 Transcription Factor--metabolism
Splenomegaly--metabolism
Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805. [electronic resource] - Molecular cancer therapeutics Jul 2010 - 1945-55 p. digital
Publication Type: Journal Article
1538-8514
10.1158/1535-7163.MCT-10-0053 doi
Adenosine Triphosphate--pharmacology
Animals
Apoptosis--drug effects
Cell Line
Cell Line, Tumor
Cell Proliferation--drug effects
Erythropoiesis--drug effects
Humans
Janus Kinase 2--antagonists & inhibitors
K562 Cells
Mice
Mice, Inbred BALB C
Mice, SCID
Models, Molecular
Molecular Structure
Mutation
Phosphorylation--drug effects
Polycythemia--metabolism
Protein Structure, Tertiary
Quinoxalines--chemistry
Rats
STAT5 Transcription Factor--metabolism
Splenomegaly--metabolism