Purified E255L mutant SERCA1a and purified PfATP6 are sensitive to SERCA-type inhibitors but insensitive to artemisinins.
Cardi, Delphine
Purified E255L mutant SERCA1a and purified PfATP6 are sensitive to SERCA-type inhibitors but insensitive to artemisinins. [electronic resource] - The Journal of biological chemistry Aug 2010 - 26406-16 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1083-351X
10.1074/jbc.M109.090340 doi
Animals
Antimalarials
Artemisinins--pharmacology
COS Cells
Calcium-Transporting ATPases--drug effects
Chlorocebus aethiops
Enzyme Inhibitors--pharmacology
Mutant Proteins
Mutation, Missense
Rabbits
Saccharomyces cerevisiae
Sarcoplasmic Reticulum Calcium-Transporting ATPases--antagonists & inhibitors
Purified E255L mutant SERCA1a and purified PfATP6 are sensitive to SERCA-type inhibitors but insensitive to artemisinins. [electronic resource] - The Journal of biological chemistry Aug 2010 - 26406-16 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1083-351X
10.1074/jbc.M109.090340 doi
Animals
Antimalarials
Artemisinins--pharmacology
COS Cells
Calcium-Transporting ATPases--drug effects
Chlorocebus aethiops
Enzyme Inhibitors--pharmacology
Mutant Proteins
Mutation, Missense
Rabbits
Saccharomyces cerevisiae
Sarcoplasmic Reticulum Calcium-Transporting ATPases--antagonists & inhibitors