Organic cation transporters modulate the uptake and cytotoxicity of picoplatin, a third-generation platinum analogue.
More, Swati S
Organic cation transporters modulate the uptake and cytotoxicity of picoplatin, a third-generation platinum analogue. [electronic resource] - Molecular cancer therapeutics Apr 2010 - 1058-69 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1538-8514
10.1158/1535-7163.MCT-09-1084 doi
Animals
Cell Death--drug effects
Cell Line, Tumor
Cimetidine--pharmacology
DNA Adducts--metabolism
Gene Expression Regulation, Neoplastic--drug effects
Humans
Lung Neoplasms--genetics
Mice
Organic Cation Transport Proteins--antagonists & inhibitors
Platinum Compounds--pharmacokinetics
Polymorphism, Single Nucleotide--genetics
Tissue Distribution--drug effects
Xenograft Model Antitumor Assays
Organic cation transporters modulate the uptake and cytotoxicity of picoplatin, a third-generation platinum analogue. [electronic resource] - Molecular cancer therapeutics Apr 2010 - 1058-69 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1538-8514
10.1158/1535-7163.MCT-09-1084 doi
Animals
Cell Death--drug effects
Cell Line, Tumor
Cimetidine--pharmacology
DNA Adducts--metabolism
Gene Expression Regulation, Neoplastic--drug effects
Humans
Lung Neoplasms--genetics
Mice
Organic Cation Transport Proteins--antagonists & inhibitors
Platinum Compounds--pharmacokinetics
Polymorphism, Single Nucleotide--genetics
Tissue Distribution--drug effects
Xenograft Model Antitumor Assays