Evolving carbapenemases: can medicinal chemists advance one step ahead of the coming storm?

Oelschlaeger, Peter

Evolving carbapenemases: can medicinal chemists advance one step ahead of the coming storm? [electronic resource] - Journal of medicinal chemistry Apr 2010 - 3013-27 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm9012938 doi


Algorithms
Anti-Bacterial Agents--chemistry
Bacterial Proteins--antagonists & inhibitors
Carbapenems--chemistry
Crystallography, X-Ray
Databases, Factual
Drug Design
Drug Resistance, Multiple, Bacterial
Klebsiella pneumoniae--enzymology
Metalloproteins--antagonists & inhibitors
Models, Molecular
Mutation
Protein Conformation
Substrate Specificity
beta-Lactamase Inhibitors
beta-Lactamases--chemistry