Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation.
Kuck, Dirk
Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation. [electronic resource] - Bioorganic & medicinal chemistry Jan 2010 - 822-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2009.11.050 doi
Cloning, Molecular
Crystallography, X-Ray
DNA (Cytosine-5-)-Methyltransferase 1
DNA (Cytosine-5-)-Methyltransferases--antagonists & inhibitors
Dose-Response Relationship, Drug
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemistry
Humans
Models, Molecular
Structure-Activity Relationship
DNA Methyltransferase 3B
Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation. [electronic resource] - Bioorganic & medicinal chemistry Jan 2010 - 822-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2009.11.050 doi
Cloning, Molecular
Crystallography, X-Ray
DNA (Cytosine-5-)-Methyltransferase 1
DNA (Cytosine-5-)-Methyltransferases--antagonists & inhibitors
Dose-Response Relationship, Drug
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemistry
Humans
Models, Molecular
Structure-Activity Relationship
DNA Methyltransferase 3B