Biaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part I.
Trova, Michael P
Biaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part I. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2009 - 6608-12 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.10.025 doi
Antineoplastic Agents--chemical synthesis
Cell Proliferation--drug effects
Cyclin-Dependent Kinases--antagonists & inhibitors
Drug Design
Drug Screening Assays, Antitumor
HeLa Cells
Humans
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Purines--chemical synthesis
Roscovitine
Stereoisomerism
Structure-Activity Relationship
Biaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part I. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2009 - 6608-12 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.10.025 doi
Antineoplastic Agents--chemical synthesis
Cell Proliferation--drug effects
Cyclin-Dependent Kinases--antagonists & inhibitors
Drug Design
Drug Screening Assays, Antitumor
HeLa Cells
Humans
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Purines--chemical synthesis
Roscovitine
Stereoisomerism
Structure-Activity Relationship