Inhibitors of bacterial N-succinyl-L,L-diaminopimelic acid desuccinylase (DapE) and demonstration of in vitro antimicrobial activity.
Gillner, Danuta
Inhibitors of bacterial N-succinyl-L,L-diaminopimelic acid desuccinylase (DapE) and demonstration of in vitro antimicrobial activity. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2009 - 6350-2 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
1464-3405
10.1016/j.bmcl.2009.09.077 doi
Amidohydrolases--antagonists & inhibitors
Amino Acid Sequence
Anti-Bacterial Agents--pharmacology
Binding Sites
Diaminopimelic Acid--metabolism
Enzyme Inhibitors--pharmacology
Escherichia coli--drug effects
Haemophilus influenzae--drug effects
Microbial Sensitivity Tests
Mutagenesis, Site-Directed
Substrate Specificity
Inhibitors of bacterial N-succinyl-L,L-diaminopimelic acid desuccinylase (DapE) and demonstration of in vitro antimicrobial activity. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2009 - 6350-2 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
1464-3405
10.1016/j.bmcl.2009.09.077 doi
Amidohydrolases--antagonists & inhibitors
Amino Acid Sequence
Anti-Bacterial Agents--pharmacology
Binding Sites
Diaminopimelic Acid--metabolism
Enzyme Inhibitors--pharmacology
Escherichia coli--drug effects
Haemophilus influenzae--drug effects
Microbial Sensitivity Tests
Mutagenesis, Site-Directed
Substrate Specificity