Pyrazole NNRTIs 1: design and initial optimisation of a novel template.

Mowbray, Charles E

Pyrazole NNRTIs 1: design and initial optimisation of a novel template. [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2009 - 5599-602 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2009.08.039 doi


Anti-HIV Agents--chemical synthesis
Drug Design
HIV Reverse Transcriptase--antagonists & inhibitors
Humans
Microsomes, Liver--metabolism
Pyrazoles--chemical synthesis
Reverse Transcriptase Inhibitors--chemical synthesis
Structure-Activity Relationship