Pharmacological characterization of INCB3344, a small molecule antagonist of human CCR2.
Shin, Niu
Pharmacological characterization of INCB3344, a small molecule antagonist of human CCR2. [electronic resource] - Biochemical and biophysical research communications Sep 2009 - 251-5 p. digital
Publication Type: Journal Article
1090-2104
10.1016/j.bbrc.2009.06.135 doi
Biological Assay
Cells, Cultured
Chemokine CCL2--metabolism
Chemotaxis
Extracellular Signal-Regulated MAP Kinases--metabolism
Flow Cytometry--methods
Humans
Leukocytes, Mononuclear--drug effects
Phosphorylation
Pyrrolidines--metabolism
Receptors, CCR2--antagonists & inhibitors
Pharmacological characterization of INCB3344, a small molecule antagonist of human CCR2. [electronic resource] - Biochemical and biophysical research communications Sep 2009 - 251-5 p. digital
Publication Type: Journal Article
1090-2104
10.1016/j.bbrc.2009.06.135 doi
Biological Assay
Cells, Cultured
Chemokine CCL2--metabolism
Chemotaxis
Extracellular Signal-Regulated MAP Kinases--metabolism
Flow Cytometry--methods
Humans
Leukocytes, Mononuclear--drug effects
Phosphorylation
Pyrrolidines--metabolism
Receptors, CCR2--antagonists & inhibitors