Development and applications of a broad-coverage, TR-FRET-based kinase binding assay platform.

Lebakken, Connie S

Development and applications of a broad-coverage, TR-FRET-based kinase binding assay platform. [electronic resource] - Journal of biomolecular screening Sep 2009 - 924-35 p. digital

Publication Type: Evaluation Study; Journal Article

1552-454X

10.1177/1087057109339207 doi


Animals
Cells, Cultured
Cyclic AMP--analogs & derivatives
Cyclin-Dependent Kinases--antagonists & inhibitors
Drug Evaluation, Preclinical--instrumentation
Fluorescence Resonance Energy Transfer--instrumentation
Fluorescent Dyes--chemistry
HeLa Cells
High-Throughput Screening Assays--instrumentation
Humans
Models, Biological
Phosphotransferases--antagonists & inhibitors
Protein Binding
Protein Kinase Inhibitors--analysis
Proto-Oncogene Proteins B-raf--antagonists & inhibitors
Staurosporine--chemistry
p38 Mitogen-Activated Protein Kinases--antagonists & inhibitors