Optimization of 5-phenyl-3-pyridinecarbonitriles as PKCtheta inhibitors.

Boschelli, Diane H

Optimization of 5-phenyl-3-pyridinecarbonitriles as PKCtheta inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Jul 2009 - 3623-6 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2009.04.126 doi


Animals
Indoles--chemical synthesis
Isoenzymes--antagonists & inhibitors
Mice
Nitriles--chemical synthesis
Protein Kinase C--antagonists & inhibitors
Protein Kinase C-theta
Protein Kinase Inhibitors--chemical synthesis
Pyridines--chemical synthesis
Structure-Activity Relationship