Arylphthalazines as potent, and orally bioavailable inhibitors of VEGFR-2.

Duncton, Matthew A J

Arylphthalazines as potent, and orally bioavailable inhibitors of VEGFR-2. [electronic resource] - Bioorganic & medicinal chemistry Jan 2009 - 731-40 p. digital

Publication Type: Journal Article

1464-3391

10.1016/j.bmc.2008.11.049 doi


Administration, Oral
Animals
Biological Availability
Female
Isoquinolines--chemical synthesis
Mice
Mice, Inbred Strains
Phthalazines--administration & dosage
Piperidines
Quinazolines
Vascular Endothelial Growth Factor Receptor-1--antagonists & inhibitors
Vascular Endothelial Growth Factor Receptor-2--antagonists & inhibitors