Discovery and characterization of novel allosteric potentiators of M1 muscarinic receptors reveals multiple modes of activity.

Marlo, Joy E

Discovery and characterization of novel allosteric potentiators of M1 muscarinic receptors reveals multiple modes of activity. [electronic resource] - Molecular pharmacology Mar 2009 - 577-88 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1521-0111

10.1124/mol.108.052886 doi


Allosteric Regulation--drug effects
Animals
Binding, Competitive--drug effects
CHO Cells
Cells, Cultured
Cricetinae
Cricetulus
Dose-Response Relationship, Drug
Humans
Muscarinic Agonists--chemistry
Rats
Receptor, Muscarinic M1--agonists