Structure-based design of a novel class of potent inhibitors of InhA, the enoyl acyl carrier protein reductase from Mycobacterium tuberculosis: a computer modelling approach.

Subba Rao, Gita

Structure-based design of a novel class of potent inhibitors of InhA, the enoyl acyl carrier protein reductase from Mycobacterium tuberculosis: a computer modelling approach. [electronic resource] - Chemical biology & drug design Nov 2008 - 444-9 p. digital

Publication Type: Journal Article

1747-0285

10.1111/j.1747-0285.2008.00722.x doi


Antitubercular Agents--chemistry
Bacterial Proteins--antagonists & inhibitors
Computer Simulation
Drug Design
Enoyl-(Acyl-Carrier-Protein) Reductase (NADH)--antagonists & inhibitors
Mycobacterium tuberculosis--enzymology
Oxidoreductases--antagonists & inhibitors
Peptides--chemistry
Protein Structure, Tertiary
Structure-Activity Relationship