Dihydropyrrole[2,3-d]pyridine derivatives as novel corticotropin-releasing factor-1 antagonists: mapping of the receptor binding pocket by in silico docking studies.

Di Fabio, Romano

Dihydropyrrole[2,3-d]pyridine derivatives as novel corticotropin-releasing factor-1 antagonists: mapping of the receptor binding pocket by in silico docking studies. [electronic resource] - Journal of medicinal chemistry Nov 2008 - 7273-86 p. digital

Publication Type: Journal Article

1520-4804

10.1021/jm800743q doi


Animals
Binding Sites
CHO Cells
Computer Simulation
Cricetinae
Cricetulus
Drug Design
Ligands
Molecular Structure
Pyridines--chemical synthesis
Pyrroles--chemical synthesis
Quantitative Structure-Activity Relationship
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Stereoisomerism
CRF Receptor, Type 1