Pimelic diphenylamide 106 is a slow, tight-binding inhibitor of class I histone deacetylases.
Chou, C James
Pimelic diphenylamide 106 is a slow, tight-binding inhibitor of class I histone deacetylases. [electronic resource] - The Journal of biological chemistry Dec 2008 - 35402-9 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
0021-9258
10.1074/jbc.M807045200 doi
Animals
Disease Models, Animal
Enzyme Inhibitors--chemistry
Friedreich Ataxia--drug therapy
Histone Deacetylase Inhibitors
Histone Deacetylases--metabolism
Humans
Huntington Disease--drug therapy
Isoenzymes--antagonists & inhibitors
Kinetics
Mice
Neoplasm Proteins--antagonists & inhibitors
Neoplasms--drug therapy
Pimelic Acids--chemistry
Pimelic diphenylamide 106 is a slow, tight-binding inhibitor of class I histone deacetylases. [electronic resource] - The Journal of biological chemistry Dec 2008 - 35402-9 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
0021-9258
10.1074/jbc.M807045200 doi
Animals
Disease Models, Animal
Enzyme Inhibitors--chemistry
Friedreich Ataxia--drug therapy
Histone Deacetylase Inhibitors
Histone Deacetylases--metabolism
Humans
Huntington Disease--drug therapy
Isoenzymes--antagonists & inhibitors
Kinetics
Mice
Neoplasm Proteins--antagonists & inhibitors
Neoplasms--drug therapy
Pimelic Acids--chemistry