Kinase array design, back to front: biaryl amides.

Baldwin, Ian

Kinase array design, back to front: biaryl amides. [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2008 - 5285-9 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2008.08.051 doi


Adenosine Triphosphate--chemistry
Amides--chemical synthesis
Animals
Combinatorial Chemistry Techniques
Crystallography, X-Ray
Heterocyclic Compounds, 1-Ring--chemical synthesis
Inhibitory Concentration 50
Mitogen-Activated Protein Kinase 14--antagonists & inhibitors
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Rats
Structure-Activity Relationship