Baicalin, a prodrug able to reach the CNS, is a prolyl oligopeptidase inhibitor.

Tarragó, Teresa

Baicalin, a prodrug able to reach the CNS, is a prolyl oligopeptidase inhibitor. [electronic resource] - Bioorganic & medicinal chemistry Aug 2008 - 7516-24 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2008.04.067 doi


Dose-Response Relationship, Drug
Enzyme Inhibitors--chemistry
Flavanones--chemistry
Flavonoids--chemistry
Prolyl Oligopeptidases
Serine Endopeptidases--metabolism
Structure-Activity Relationship