Bioisosteric phentolamine analogs as selective human alpha(2)- versus alpha(1)-adrenoceptor ligands.

Bavadekar, Supriya A

Bioisosteric phentolamine analogs as selective human alpha(2)- versus alpha(1)-adrenoceptor ligands. [electronic resource] - European journal of pharmacology Aug 2008 - 53-60 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.

0014-2999

10.1016/j.ejphar.2008.05.027 doi


Animals
CHO Cells
Cricetinae
Cricetulus
Cyclic AMP--pharmacology
Humans
Luciferases--genetics
Phentolamine--analogs & derivatives
Radioligand Assay
Receptors, Adrenergic, alpha-1--metabolism
Receptors, Adrenergic, alpha-2--metabolism
Response Elements
Structure-Activity Relationship