In vitro evaluation of photosensitivity risk related to genetic polymorphisms of human ABC transporter ABCG2 and inhibition by drugs.

Tamura, Ai

In vitro evaluation of photosensitivity risk related to genetic polymorphisms of human ABC transporter ABCG2 and inhibition by drugs. [electronic resource] - Drug metabolism and pharmacokinetics Dec 2007 - 428-40 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1347-4367

10.2133/dmpk.22.428 doi


ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--antagonists & inhibitors
Animals
Benzamides
Cell Line
Cell Survival--drug effects
Chlorophyll--analogs & derivatives
Dose-Response Relationship, Drug
Drug Interactions
Homeostasis
Humans
Imatinib Mesylate
Inhibitory Concentration 50
Insecta
Light
Membrane Transport Modulators--toxicity
Microscopy, Fluorescence
Neoplasm Proteins--antagonists & inhibitors
Novobiocin--toxicity
Photosensitivity Disorders--chemically induced
Photosensitizing Agents--metabolism
Piperazines--toxicity
Polymorphism, Single Nucleotide
Porphyrins--metabolism
Pyrimidines--toxicity
Quercetin--pharmacology
Risk Assessment
Transfection