Modulation of P-glycoprotein-mediated multidrug resistance by acceleration of passive drug permeation across the plasma membrane.
Regev, Ronit
Modulation of P-glycoprotein-mediated multidrug resistance by acceleration of passive drug permeation across the plasma membrane. [electronic resource] - The FEBS journal Dec 2007 - 6204-14 p. digital
Publication Type: Journal Article
1742-464X
10.1111/j.1742-4658.2007.06140.x doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Acceleration
Anesthetics--pharmacology
Antibiotics, Antineoplastic--metabolism
Biological Transport--drug effects
Calcium Channel Blockers--metabolism
Cell Membrane--drug effects
Cell Membrane Permeability
Daunorubicin--metabolism
Dose-Response Relationship, Drug
Drug Resistance, Multiple
Drug Resistance, Neoplasm
Drug Synergism
Excipients--pharmacology
Fluorescence Polarization
Fluorescent Dyes--pharmacokinetics
Humans
K562 Cells
Membrane Fluidity--drug effects
Rhodamines--pharmacokinetics
Surface-Active Agents--pharmacology
Verapamil--metabolism
Modulation of P-glycoprotein-mediated multidrug resistance by acceleration of passive drug permeation across the plasma membrane. [electronic resource] - The FEBS journal Dec 2007 - 6204-14 p. digital
Publication Type: Journal Article
1742-464X
10.1111/j.1742-4658.2007.06140.x doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Acceleration
Anesthetics--pharmacology
Antibiotics, Antineoplastic--metabolism
Biological Transport--drug effects
Calcium Channel Blockers--metabolism
Cell Membrane--drug effects
Cell Membrane Permeability
Daunorubicin--metabolism
Dose-Response Relationship, Drug
Drug Resistance, Multiple
Drug Resistance, Neoplasm
Drug Synergism
Excipients--pharmacology
Fluorescence Polarization
Fluorescent Dyes--pharmacokinetics
Humans
K562 Cells
Membrane Fluidity--drug effects
Rhodamines--pharmacokinetics
Surface-Active Agents--pharmacology
Verapamil--metabolism