Identification and characterization of a selective peroxisome proliferator-activated receptor beta/delta (NR1C2) antagonist.

Shearer, Barry G

Identification and characterization of a selective peroxisome proliferator-activated receptor beta/delta (NR1C2) antagonist. [electronic resource] - Molecular endocrinology (Baltimore, Md.) Feb 2008 - 523-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0888-8809

10.1210/me.2007-0190 doi


Cells, Cultured
Chromatin Immunoprecipitation
Dose-Response Relationship, Drug
Fatty Acids--metabolism
Fluorescence Resonance Energy Transfer
Gene Expression Regulation--drug effects
Humans
Ligands
Molecular Structure
Muscle, Skeletal--cytology
Oxidation-Reduction--drug effects
PPAR delta--antagonists & inhibitors
PPAR-beta--antagonists & inhibitors
Sulfones--chemistry
Thiazoles--chemistry
Thiophenes--chemistry