Synthesis and in-vitro biological activity of macrocyclic urea Chk1 inhibitors.
Li, Gaoquan
Synthesis and in-vitro biological activity of macrocyclic urea Chk1 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2007 - 6499-504 p. digital
Publication Type: Comparative Study; Journal Article
1464-3405
10.1016/j.bmcl.2007.09.088 doi
Cell Line, Tumor
Checkpoint Kinase 1
HeLa Cells
Humans
Macrocyclic Compounds--chemical synthesis
Protein Kinase Inhibitors--chemical synthesis
Protein Kinases--metabolism
Structure-Activity Relationship
Urea--chemical synthesis
Synthesis and in-vitro biological activity of macrocyclic urea Chk1 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2007 - 6499-504 p. digital
Publication Type: Comparative Study; Journal Article
1464-3405
10.1016/j.bmcl.2007.09.088 doi
Cell Line, Tumor
Checkpoint Kinase 1
HeLa Cells
Humans
Macrocyclic Compounds--chemical synthesis
Protein Kinase Inhibitors--chemical synthesis
Protein Kinases--metabolism
Structure-Activity Relationship
Urea--chemical synthesis