Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors.

Brnardic, Edward J

Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2007 - 5989-94 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2007.07.051 doi


Checkpoint Kinase 1
Crystallography, X-Ray
Models, Molecular
Protein Kinase Inhibitors--chemistry
Protein Kinases--drug effects
Quinolones--chemistry
Structure-Activity Relationship