Design and synthesis of benzoazepinone-derived cyclic malonamides and aminoamides as potent gamma-secretase inhibitors.

Yang, Michael G

Design and synthesis of benzoazepinone-derived cyclic malonamides and aminoamides as potent gamma-secretase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Jul 2007 - 3910-5 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2007.04.102 doi


Amides--pharmacology
Amyloid Precursor Protein Secretases--antagonists & inhibitors
Azepines--chemical synthesis
Cyclization
Models, Molecular
Structure-Activity Relationship