Cholesterol potentiates ABCG2 activity in a heterologous expression system: improved in vitro model to study function of human ABCG2.
Pál, A
Cholesterol potentiates ABCG2 activity in a heterologous expression system: improved in vitro model to study function of human ABCG2. [electronic resource] - The Journal of pharmacology and experimental therapeutics Jun 2007 - 1085-94 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-3565
10.1124/jpet.106.119289 doi
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--genetics
Adenosine Triphosphatases--metabolism
Animals
Baculoviridae--genetics
Benzimidazoles--metabolism
Biological Transport, Active--drug effects
Cell Line
Cell Membrane--metabolism
Cholesterol--pharmacology
Estrone--analogs & derivatives
Glycosylation
Humans
Kinetics
Methotrexate--metabolism
Neoplasm Proteins--genetics
Peptide-N4-(N-acetyl-beta-glucosaminyl) Asparagine Amidase--metabolism
Pharmaceutical Preparations--metabolism
Prazosin--metabolism
Spodoptera
Sulfasalazine--metabolism
Topotecan--metabolism
Cholesterol potentiates ABCG2 activity in a heterologous expression system: improved in vitro model to study function of human ABCG2. [electronic resource] - The Journal of pharmacology and experimental therapeutics Jun 2007 - 1085-94 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-3565
10.1124/jpet.106.119289 doi
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--genetics
Adenosine Triphosphatases--metabolism
Animals
Baculoviridae--genetics
Benzimidazoles--metabolism
Biological Transport, Active--drug effects
Cell Line
Cell Membrane--metabolism
Cholesterol--pharmacology
Estrone--analogs & derivatives
Glycosylation
Humans
Kinetics
Methotrexate--metabolism
Neoplasm Proteins--genetics
Peptide-N4-(N-acetyl-beta-glucosaminyl) Asparagine Amidase--metabolism
Pharmaceutical Preparations--metabolism
Prazosin--metabolism
Spodoptera
Sulfasalazine--metabolism
Topotecan--metabolism