Additional evidence for functional subclassification of alpha-2 adrenoceptors based on a new selective antagonist, SK&F 104856.

Hieble, J P

Additional evidence for functional subclassification of alpha-2 adrenoceptors based on a new selective antagonist, SK&F 104856. [electronic resource] - The Journal of pharmacology and experimental therapeutics Nov 1991 - 643-52 p. digital

Publication Type: Journal Article

0022-3565


Adrenergic alpha-Agonists--pharmacology
Adrenergic alpha-Antagonists--metabolism
Animals
Atrial Function
Benzazepines--pharmacology
Binding, Competitive
Brimonidine Tartrate
Dogs
Electric Stimulation
Female
Guinea Pigs
Heart Atria--drug effects
Humans
In Vitro Techniques
Male
Muscle Contraction--drug effects
Muscle, Smooth, Vascular--drug effects
Norepinephrine--physiology
Quinoxalines--pharmacology
Rabbits
Rats
Rats, Inbred Strains
Receptors, Adrenergic, alpha--classification
Serotonin--physiology
Synaptic Transmission--drug effects
Tritium
Vas Deferens--drug effects