Discovery of tetralin ureas as potent melanin concentrating hormone 1 receptor antagonists.

Guo, Tao

Discovery of tetralin ureas as potent melanin concentrating hormone 1 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2007 - 1718-21 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2006.12.080 doi


Animals
Binding, Competitive--drug effects
CHO Cells
Cricetinae
Cricetulus
Drug Design
Humans
Mice
Mice, Knockout
Rats
Receptors, Somatostatin--antagonists & inhibitors
Structure-Activity Relationship
Tetrahydronaphthalenes--chemical synthesis
Tissue Distribution
Urea--analogs & derivatives