Allosteric and orthosteric binding modes of two nonpeptide human gonadotropin-releasing hormone receptor antagonists.

Sullivan, Susan K

Allosteric and orthosteric binding modes of two nonpeptide human gonadotropin-releasing hormone receptor antagonists. [electronic resource] - Biochemistry Dec 2006 - 15327-37 p. digital

Publication Type: Journal Article

1520-4995

10.1021/bi0617097 doi


Allosteric Regulation--genetics
Animals
Binding Sites--genetics
Binding, Competitive--genetics
COS Cells
Cell Line, Tumor
Chlorocebus aethiops
Furans--metabolism
Hormone Antagonists--metabolism
Humans
Inhibitory Concentration 50
Mutagenesis, Site-Directed
Radioligand Assay
Rats
Receptors, LHRH--agonists
Stereoisomerism
Thymine--analogs & derivatives