Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists.
Meyers, Kenneth M
Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2007 - 657-61 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.10.096 doi
Caco-2 Cells
Humans
Indicators and Reagents
Models, Molecular
Molecular Conformation
Piperazines--chemical synthesis
Pyrazoles--chemical synthesis
Pyrroles--chemical synthesis
Radioligand Assay
Receptor, Serotonin, 5-HT2C--drug effects
Receptors, Somatostatin--antagonists & inhibitors
Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2007 - 657-61 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.10.096 doi
Caco-2 Cells
Humans
Indicators and Reagents
Models, Molecular
Molecular Conformation
Piperazines--chemical synthesis
Pyrazoles--chemical synthesis
Pyrroles--chemical synthesis
Radioligand Assay
Receptor, Serotonin, 5-HT2C--drug effects
Receptors, Somatostatin--antagonists & inhibitors