Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition.
Tian, Gaochao
Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition. [electronic resource] - Molecular pharmacology Mar 2007 - 902-11 p. digital
Publication Type: Journal Article
0026-895X
10.1124/mol.106.029868 doi
Animals
Binding, Competitive
CHO Cells
Calcium--metabolism
Cricetinae
Cricetulus
Kinetics
Neurokinin B--analogs & derivatives
Piperidines--metabolism
Quinolines--metabolism
Receptors, Neurokinin-3--antagonists & inhibitors
Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition. [electronic resource] - Molecular pharmacology Mar 2007 - 902-11 p. digital
Publication Type: Journal Article
0026-895X
10.1124/mol.106.029868 doi
Animals
Binding, Competitive
CHO Cells
Calcium--metabolism
Cricetinae
Cricetulus
Kinetics
Neurokinin B--analogs & derivatives
Piperidines--metabolism
Quinolines--metabolism
Receptors, Neurokinin-3--antagonists & inhibitors